SCHEMBL20125129

SCHEMBL20125129

COc1ccc(C)cc1NC(=O)CN1CCOCC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.70
LMNA P02545 6/20 0.70
MAPT P10636 3/20 0.69
NPSR1 Q6W5P4 2/20 0.69
KMT2A Q03164 8/20 0.69
MEN1 O00255 6/20 0.69
SMN1; SMN2 Q16637 3/20 0.69
TP53 P04637 1/20 0.69
ALOX15 P16050 1/20 0.65
TSHR P16473 4/20 0.64
KDM4E B2RXH2 1/20 0.64
THRB P10828 1/20 0.64
MAPK1 P28482 2/20 0.63
USP2 O75604 1/20 0.63
GAA P10253 3/20 0.62
HSD17B10 Q99714 1/20 0.62
CYP1A2 P05177 1/20 0.61
CYP3A4 P08684 1/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16097533 0.87 RAD52 (0.80) ALDH1A1LMNAMAPTKMT2AMEN1
SCHEMBL16097710 0.86 MAPT (0.69) ALDH1A1LMNAMAPTKMT2AMEN1
SCHEMBL16097706 0.86 ALDH1A1 (0.76) ALDH1A1LMNAMAPTKMT2AMEN1
SCHEMBL15829432 0.85 MAPT (0.65) ALDH1A1LMNAMAPTNPSR1KMT2A
SCHEMBL1643927 0.84 ALDH1A1 (0.76) ALDH1A1LMNAMAPTNPSR1KMT2A
SCHEMBL16098653 0.83 KMT2A (0.84) ALDH1A1LMNAMAPTKMT2AMEN1
SCHEMBL5506340 0.80 ALDH1A1 (0.57) ALDH1A1LMNAMAPTNPSR1KMT2A
SCHEMBL16097379 0.80 WNT3A (0.69) ALDH1A1LMNAMAPTSMN1; SMN2ALOX15
SCHEMBL21722001 0.80 MAPT (0.64) ALDH1A1LMNAMAPTKMT2AMEN1
SCHEMBL27000659 0.80 KDM4E (0.69) ALDH1A1LMNAMAPTKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3318557-A2 QUINOLONE COMPOUND Otsuka Pharmaceutical Co., Ltd. (JP) 2018-05-09 EP disclosed