SCHEMBL20125477

SCHEMBL20125477

O=Cc1ccnc2cc(COc3ccccc3)[nH]c12

nearest known ligand 0.65

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 2/20 0.65
KDM4C Q9H3R0 15/20 0.52
KDM5B Q9UGL1 10/20 0.52
KDM5A P29375 9/20 0.52
NPY5R Q15761 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20125409 0.82 KDM5B (0.65) KDM4AKDM4CKDM5BKDM5A
SCHEMBL20125266 0.82 KDM5B (0.61) KDM4AKDM4CKDM5BKDM5A
SCHEMBL16157388 0.79 KDM4A (1.00) KDM4AKDM4CKDM5BKDM5A
SCHEMBL20125363 0.77 KDM5B (0.60) KDM4AKDM4CKDM5BKDM5A
SCHEMBL20125343 0.74 KDM4C (0.49) KDM4AKDM4CKDM5BKDM5A
SCHEMBL20125489 0.72 KDM5B (0.63) KDM4AKDM4CKDM5BKDM5A
SCHEMBL20125359 0.71 KDM5B (0.66) KDM4AKDM4CKDM5BKDM5A
SCHEMBL20125267 0.70 KDM5B (0.65) KDM4AKDM4CKDM5BKDM5ANPY5R
SCHEMBL20125365 0.70 KDM5A (0.56) KDM4AKDM4CKDM5BKDM5A
SCHEMBL16150315 0.69 KDM4C (0.69) KDM4AKDM4CKDM5BKDM5ANPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968282-B1 HISTONE DEMENTHYLASE INHIBITORS CELGENE QUANTICEL RES INC (US) 2018-05-09 EP disclosed