SCHEMBL2012817

SCHEMBL2012817

CNC(=O)c1cc(F)cc(-c2c(CCNc3ncnc4[nH]cnc34)cc(Cl)c3ccnnc23)c1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.42
MAP4K4 O95819 3/20 0.37
BCL2 P10415 1/20 0.36
CDK1 P06493 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012486 0.90 PIK3CD (0.46) PIK3CDBCL2
SCHEMBL2016865 0.84 PIK3CD (0.56) PIK3CDMAP4K4BCL2
SCHEMBL2012816 0.83 PIK3CD (0.59) PIK3CDMAP4K4BCL2
Trifluoroacetic Acid SCHEMBL2050998 0.82 PIK3CD (0.40) PIK3CDBCL2
SCHEMBL2017997 0.82 PIK3CD (0.39) PIK3CDBCL2
Trifluoroacetic Acid SCHEMBL2052496 0.80 PIK3CD (0.35) PIK3CD
SCHEMBL2051059 0.80 PIK3CD (0.53) PIK3CDMAP4K4BCL2
SCHEMBL2050306 0.79 PIK3CD (0.42) PIK3CDBCL2
SCHEMBL2052089 0.76 PIK3CD (0.48) PIK3CDMAP4K4BCL2
SCHEMBL2016719 0.76 PIK3CD (0.47) PIK3CDMAP4K4BCL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO claimed
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed