SCHEMBL2012874

SCHEMBL2012874

CN(C(=O)c1cc(Cl)cc2cccnc12)C(CCNC(=O)c1cccn1C)Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.58
HCRTR2 O43614 2/20 0.58
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
OPRM1 P35372 1/20 0.36
STING1 Q86WV6 1/20 0.36
PADI4 Q9UM07 3/20 0.36
EGLN1 Q9GZT9 2/20 0.35
HRH3 Q9Y5N1 2/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
PYGL P06737 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012875 1.00 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AOPRM1
SCHEMBL2010789 0.91 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2015844 0.90 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2012888 0.90 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2015171 0.89 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AEGLN1
SCHEMBL2015191 0.83 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AOPRM1
SCHEMBL2053648 0.82 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2016530 0.82 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9APADI4
SCHEMBL2013533 0.82 HCRTR1 (0.60) HCRTR1HCRTR2NPC1RAB9AOPRM1
SCHEMBL2054405 0.82 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9APADI4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed