SCHEMBL2015171

SCHEMBL2015171

COc1cc(C(=O)N(C)C(CCNC(=O)c2cccn2C)Cc2ccccc2)c2ncccc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.60
HCRTR2 O43614 2/20 0.60
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 2/20 0.39
KMT2A Q03164 3/20 0.38
EGLN1 Q9GZT9 2/20 0.38
MEN1 O00255 2/20 0.38
KDM4E B2RXH2 1/20 0.37
THRB P10828 1/20 0.37
CASP1 P29466 1/20 0.37
RAD52 P43351 1/20 0.37
CASP7 P55210 1/20 0.37
CASP6 P55212 1/20 0.37
CASP8 Q14790 1/20 0.37
HDAC1 Q13547 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
HRH3 Q9Y5N1 2/20 0.36
TMEM97 Q5BJF2 1/20 0.36
SIGMAR1 Q99720 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2010789 0.90 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AEGLN1
SCHEMBL2013457 0.89 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL2054419 0.89 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AALDH1A1
SCHEMBL2012875 0.89 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AEGLN1
SCHEMBL2012874 0.89 HCRTR1 (0.58) HCRTR1HCRTR2NPC1RAB9AEGLN1
SCHEMBL2015844 0.88 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AKMT2A
SCHEMBL2012888 0.88 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AKMT2A
SCHEMBL2015046 0.85 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9AKDM4E
SCHEMBL2054405 0.85 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9AKDM4E
SCHEMBL2054013 0.85 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed