SCHEMBL2013215

SCHEMBL2013215

Cc1cc(F)c(F)cc1-c1ccccc1OCc1cccc(CBr)c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 5/20 0.46
PTGER1 P34995 4/20 0.43
MAOB P27338 2/20 0.43
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
BRD4 O60885 3/20 0.40
FFAR1 O14842 1/20 0.38
SGMS2 Q8NHU3 2/20 0.38
GYS1 P13807 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2012748 0.88 PTGER1 (0.48) MRGPRX4PTGER1MAOBMAPTMAPK1
SCHEMBL2012939 0.86 GYS1 (0.48) MRGPRX4PTGER1MAOBGYS1
SCHEMBL2011729 0.80 GYS1 (0.54) MAOBGYS1
SCHEMBL15309708 0.79 MAPT (0.51) MRGPRX4MAPTMAPK1TDP1L3MBTL1
SCHEMBL12600498 0.73 MRGPRX4 (0.60) MRGPRX4MAPTMAPK1TDP1L3MBTL1
SCHEMBL15309905 0.71 ABCB1 (0.50) MRGPRX4MAPTMAPK1TDP1L3MBTL1
SCHEMBL2010257 0.70 GYS1 (0.68) GYS1
SCHEMBL2013211 0.70 GYS1 (0.38) MRGPRX4MAOBMAPTMAPK1TDP1
SCHEMBL15310220 0.70 L3MBTL1 (0.46) MRGPRX4MAPTMAPK1TDP1L3MBTL1
SCHEMBL2012370 0.69 GYS1 (0.52) MAOBGYS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011067266-A1 CARBOXYLIC ACID ANALOGS AS GLYCOGEN SYNTHASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-09 WO disclosed