SCHEMBL20135971

SCHEMBL20135971

COc1cc(N)c(N)cc1C=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.65
KDM4E B2RXH2 3/20 0.65
TSHR P16473 3/20 0.65
TDP1 Q9NUW8 2/20 0.65
LMNA P02545 1/20 0.52
HPGD P15428 1/20 0.52
PRKDC P78527 2/20 0.48
MAPT P10636 2/20 0.47
ERN1 O75460 5/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
CYP3A4 P08684 2/20 0.43
HSD17B10 Q99714 2/20 0.43
ALOX15 P16050 1/20 0.43
NPC1 O15118 2/20 0.42
TLR2 O60603 1/20 0.41
TLR1 Q15399 1/20 0.41
TLR6 Q9Y2C9 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24389243 0.89 ALDH1A1 (0.57) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL31469616 0.87 ALDH1A1 (0.72) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL1570740 0.87 ALDH1A1 (0.72) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL27753912 0.87 ALDH1A1 (0.72) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL12835408 0.86 ALDH1A1 (0.59) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL10985031 0.84 ALDH1A1 (0.57) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL629627 0.84 NPC1 (0.60) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL3136850 0.84 ALDH1A1 (0.90) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL19127201 0.82 ALDH1A1 (0.53) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL10849623 0.81 ALDH1A1 (0.86) ALDH1A1KDM4ETSHRTDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2828269-B1 BORONIC ACID BEARING LIPHAGANE COMPOUNDS AS INHIBITORS OF PI3K-ALPHA AND/OR BETA COUNCIL SCIENT IND RES (IN) 2018-05-16 EP disclosed