SCHEMBL20138700

SCHEMBL20138700

Fc1ccc(Oc2ncnn2C2CC2)cc1F

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.39
TRPA1 O75762 1/20 0.37
MAP4K4 O95819 1/20 0.36
MAPK14 Q16539 1/20 0.36
ADORA1 P30542 1/20 0.35
SOS1 Q07889 1/20 0.34
BTK Q06187 4/20 0.34
PDE9A O76083 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
AXL P30530 1/20 0.32
TYRO3 Q06418 1/20 0.32
CHRM5 P08912 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20138698 0.75 ADORA1 (0.36) ALKTRPA1MAP4K4MAPK14ADORA1
SCHEMBL12826223 0.62 MAP4K4 (0.49) TRPA1MAP4K4MAPK14SOS1CYP1A2
SCHEMBL24716435 0.60 PTGS1 (0.46) SOS1FFAR4
SCHEMBL14901056 0.60 PARP10 (0.55) FFAR4
SCHEMBL28811890 0.59 MAP4K4 (0.56) TRPA1MAP4K4MAPK14SOS1
SCHEMBL29860742 0.59 MAP4K4 (0.56) TRPA1MAP4K4MAPK14SOS1
SCHEMBL29513208 0.58 CA12 (0.50) CYP1A2
SCHEMBL254529 0.58 CA12 (0.50) CYP1A2
SCHEMBL2298852 0.58 PARP10 (0.49) FFAR4
SCHEMBL4336604 0.58 SOS1 (0.56) SOS1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538516-A1 PHENOXYTRIAZOLES F. Hoffmann-La Roche AG (CH) 2019-09-18 EP disclosed
WO-2018087018-A1 PHENOXYTRIAZOLES F. HOFFMANN-LA ROCHE AG (CH) 2018-05-17 WO disclosed