SCHEMBL20138944

SCHEMBL20138944

CCOC(=O)C(F)C(=O)C1CCOCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TSHR P16473 2/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
GAA P10253 2/20 0.37
RECQL P46063 1/20 0.36
PPM1B O75688 1/20 0.35
PTPN1 P18031 1/20 0.35
PPP1CC P36873 1/20 0.35
POLB P06746 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LGMN Q99538 1/20 0.33
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19995332 0.83 PIK3CD (0.36)
SCHEMBL3605660 0.81 CYP3A4 (0.42) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL3606175 0.80 ALDH1A1 (0.41) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL16210542 0.80 ALDH1A1 (0.41) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL957454 0.80 ALDH1A1 (0.41) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL1565504 0.76 ALDH1A1 (0.46) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL72855 0.74 MAPT (0.51) ALDH1A1LMNAMAPTTSHRCYP3A4
SCHEMBL24869876 0.72 ALDH1A1 (0.59) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL3940169 0.72 TSHR (0.43) ALDH1A1LMNAMAPTHPGDRAB9A
SCHEMBL16210467 0.71 ALDH1A1 (0.36) ALDH1A1LMNAMAPTHPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11766434-B2 Pyrimidinone derivatives as CDC7 inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2023-09-26 US disclosed
US-11766434-B2 Pyrimidinone derivatives as CDC7 inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2023-09-26 US disclosed
US-11766434-B2 Pyrimidinone derivatives as CDC7 inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2023-09-26 US disclosed
CN-110088100-B Pyrimidone derivatives as CDC7 inhibitors 癌症研究科技有限公司 2023-02-17 CN disclosed
US-20220079942-A1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2022-03-17 US disclosed
US-11020396-B2 Pyrimidinone derivatives as Cdc7 inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2021-06-01 US disclosed
US-11020396-B2 Pyrimidinone derivatives as Cdc7 inhibitors CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2021-06-01 US disclosed
EP-3538523-B1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS CANCER RESEARCH TECH LTD (GB) 2021-05-19 EP disclosed
EP-3538523-B1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS CANCER RESEARCH TECH LTD (GB) 2021-05-19 EP disclosed
US-20190336502-A1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2019-11-07 US disclosed
EP-3538523-A1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS Cancer Research Technology Limited (GB) 2019-09-18 EP disclosed
WO-2018087527-A1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2018-05-17 WO disclosed
WO-2018087527-A1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2018-05-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190336502-A1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS CDC7, CDK7, CDK17 ALDH1A1 2172/4885LMNA 2422/4885MAPT 2853/4885
US-11766434-B2 Pyrimidinone derivatives as CDC7 inhibitors CDC7, CDK7, CDK17 ALDH1A1 2172/4885LMNA 2422/4885MAPT 2853/4885
US-20220079942-A1 PYRIMIDINONE DERIVATIVES AS CDC7 INHIBITORS CDC7, CDK7, CDK17 ALDH1A1 2172/4885LMNA 2422/4885MAPT 2853/4885
US-11020396-B2 Pyrimidinone derivatives as Cdc7 inhibitors CDC7, CDK7, CDK17 ALDH1A1 2172/4885LMNA 2422/4885MAPT 2853/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.