SCHEMBL20139196

SCHEMBL20139196

C[C@H]1CN(c2cc(F)cc(F)c2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 9/20 0.48
NR1H3 Q13133 8/20 0.48
MAP4K4 O95819 1/20 0.47
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
SUV39H2 Q9H5I1 2/20 0.46
GPR119 Q8TDV5 2/20 0.45
FAAH O00519 2/20 0.45
CHRM4 P08173 1/20 0.44
HDAC1 Q13547 1/20 0.43
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139239 0.89 NR1H2 (0.50) NR1H2NR1H3MAP4K4CHRM2CHRM1
SCHEMBL10210512 0.87 FAAH (0.55) NR1H2NR1H3MAP4K4SUV39H2GPR119
SCHEMBL20139215 0.87 FAAH (0.55) NR1H2NR1H3MAP4K4SUV39H2GPR119
SCHEMBL15378173 0.87 FAAH (0.55) NR1H2NR1H3MAP4K4SUV39H2GPR119
SCHEMBL30005266 0.86 SUV39H2 (0.51) NR1H2NR1H3MAP4K4SUV39H2GPR119
SCHEMBL16333806 0.85 NR1H2 (0.48) NR1H2NR1H3MAP4K4CHRM2CHRM1
SCHEMBL17385248 0.84 MAP4K4 (0.48) NR1H2NR1H3MAP4K4SUV39H2GPR119
SCHEMBL20139589 0.84 NR1H2 (0.59) NR1H2NR1H3MAP4K4CHRM2CHRM1
SCHEMBL19107116 0.83 NR1H2 (0.46) NR1H2NR1H3MAP4K4CHRM2CHRM1
SCHEMBL31046011 0.82 ROCK2 (0.53) NR1H2NR1H3MAP4K4SUV39H2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089493-A1 PYRROLE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed