SCHEMBL20140285

SCHEMBL20140285

CCOC(=O)CC(c1nc(CCCc2ccc3c(n2)N(C(=O)O)CCC3)cs1)n1nc(C)cc1C

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.34
ITGAV P06756 11/20 0.34
ITGB6 P18564 9/20 0.34
ITGA2B P08514 8/20 0.34
GAA P10253 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
POLB P06746 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29797200 0.92 PTPRB (0.32) ITGB3ITGAVITGB6ITGA2BGAA
SCHEMBL20153398 0.92 PTPRB (0.32) ITGB3ITGAVITGB6ITGA2BGAA
SCHEMBL20140236 0.84 ITGAV (0.48) ITGB3ITGAVITGB6ITGA2B
SCHEMBL21294594 0.76 ITGB3 (0.54) ITGB3ITGAVITGB6ITGA2B
SCHEMBL20139771 0.76 ITGB3 (0.54) ITGB3ITGAVITGB6ITGA2B
SCHEMBL20139769 0.76 ITGB3 (0.54) ITGB3ITGAVITGB6ITGA2B
SCHEMBL21329619 0.76 BRD4 (0.39) ITGAVITGB6GAAMAPK1
SCHEMBL20141485 0.74 ALDH1A1 (0.36) ITGB3ITGAVITGB6ITGA2BGAA
SCHEMBL20141482 0.74 ALDH1A1 (0.36) ITGB3ITGAVITGB6ITGA2BGAA
SCHEMBL20140313 0.74 NOTUM (0.40) GAAMAPK1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110167935-B 3-substituted propionic acids as alpha V integrin inhibitors 百时美施贵宝公司 2022-05-27 CN disclosed
EP-3538525-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS Bristol-Myers Squibb Company (US) 2019-09-18 EP disclosed
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed