SCHEMBL2014048

SCHEMBL2014048

NCCc1cc(Cl)c2ccccc2c1N1CCC(O)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.38
HTR2A P28223 2/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.35
HTR6 P50406 4/20 0.35
MAOB P27338 1/20 0.35
MPO P05164 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2A6 P11509 1/20 0.34
NFKB1 P19838 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
HTR2C P28335 1/20 0.34
HTR7 P34969 1/20 0.34
CTSK P43235 1/20 0.34
CYP2A13 Q16696 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2054410 0.83 TAAR1 (0.42) TAAR1HTR2AMEN1GAAKMT2A
SCHEMBL2011476 0.78 METAP2 (0.43) MEN1KMT2ACYP1A2CYP3A4CNR2
SCHEMBL2011479 0.78 METAP2 (0.43) MEN1KMT2ACYP1A2CYP3A4CNR2
SCHEMBL2018027 0.74 HTT (0.38) TAAR1MEN1KMT2ACYP1A2CYP3A4
SCHEMBL2163965 0.74 MAOB (0.35) HTR6MAOBCYP1A2CYP3A4CYP2D6
SCHEMBL2019128 0.73 METAP2 (0.44) MEN1KMT2ACYP1A2CYP3A4NFKB1
SCHEMBL2018508 0.73 KDM4E (0.43) MEN1KMT2ACYP1A2CYP3A4KDM4E
SCHEMBL2013467 0.73 SMN1; SMN2 (0.41) MEN1KMT2ACYP1A2CYP3A4KDM4E
SCHEMBL2040390 0.72 MAPT (0.40) MEN1KMT2AATMCYP1A2GRM2
SCHEMBL2014589 0.72 METAP2 (0.44) MEN1KMT2ACYP1A2CYP3A4SLC40A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011075630-A1 SUBSTITUTED FUSED ARYL AND HETEROARYL DERIVATIVES AS PI3K INHIBITORS INCYTE CORPORATION (US) 2011-06-23 WO disclosed