SCHEMBL2014073

SCHEMBL2014073

Cc1cccc(C(=O)C(N)=CNCc2ccccc2)c1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2D6 P10635 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
MEN1 O00255 2/20 0.40
KDM4E B2RXH2 1/20 0.40
AKR1B10 O60218 1/20 0.40
TRPA1 O75762 1/20 0.40
ABCB11 O95342 1/20 0.40
DHFR P00374 1/20 0.40
LMNA P02545 1/20 0.40
MPO P05164 1/20 0.40
CYP3A4 P08684 1/20 0.40
CHRM1 P11229 1/20 0.40
AKR1B1 P15121 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
AKR1C3 P42330 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2014070 1.00 KMT2A (0.40) KMT2ACYP1A2CYP2C9CYP2D6TSHR
SCHEMBL2013850 0.80 NR4A1 (0.42) KMT2ACYP1A2CYP2C9CYP2C19MEN1
SCHEMBL2013851 0.80 NR4A1 (0.42) KMT2ACYP1A2CYP2C9CYP2C19MEN1
SCHEMBL12631384 0.76 L3MBTL1 (0.50) KMT2AMEN1LMNATDP1SMN1; SMN2
SCHEMBL20344487 0.75 ADH1B (0.52) KMT2ACYP1A2CYP2C9CYP2D6TSHR
SCHEMBL7449222 0.75 ADH1B (0.52) KMT2ACYP1A2CYP2C9CYP2D6TSHR
SCHEMBL7449229 0.75 ADH1B (0.52) KMT2ACYP1A2CYP2C9CYP2D6TSHR
SCHEMBL2014206 0.73 ADH1B (0.40) KMT2ACYP1A2CYP2C9CYP2D6TSHR
SCHEMBL20344664 0.73 ADH1B (0.46) KMT2ACYP1A2CYP2C9CYP2D6TSHR
SCHEMBL19255773 0.72 SMN1; SMN2 (0.48) KMT2ACYP1A2CYP2C19MEN1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011070069-A1 PROCESS FOR PREPARATION OF MEDETOMIDINE I-TECH AB (SE) 2011-06-16 WO claimed
WO-2011070069-A1 PROCESS FOR PREPARATION OF MEDETOMIDINE I-TECH AB (SE) 2011-06-16 WO disclosed