SCHEMBL2014087

SCHEMBL2014087

Nc1nc2c(ncn2[C@@H]2O[C@H](COS)[C@@H](O)[C@H]2O)c(=O)[nH]1

nearest known ligand 0.72

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HINT1 P49773 6/20 0.72
NT5E P21589 1/20 0.72
GSK3A P49840 2/20 0.67
RPS6KA3 P51812 2/20 0.67
MAPK14 Q16539 2/20 0.67
TGM2 P21980 1/20 0.66
PNP P00491 1/20 0.64
KRAS P01116 5/20 0.60
FUT5 Q11128 1/20 0.59
HPGD P15428 1/20 0.59
IMPDH2 P12268 2/20 0.58
IMPDH1 P20839 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29211434 0.91 HINT1 (0.73) HINT1NT5EGSK3ARPS6KA3MAPK14
SCHEMBL3514472 0.91 HINT1 (0.73) HINT1NT5EGSK3ARPS6KA3MAPK14
SCHEMBL17355882 0.91 HINT1 (0.73) HINT1NT5EGSK3ARPS6KA3MAPK14
SCHEMBL3970953 0.91 HINT1 (0.73) HINT1NT5EGSK3ARPS6KA3MAPK14
2'-Beta-Methyl-Guanosine SCHEMBL15338533 0.90 HINT1 (0.75) HINT1NT5EGSK3ARPS6KA3MAPK14
2'-Beta-Methyl-Guanosine SCHEMBL14178410 0.90 HINT1 (0.75) HINT1NT5EGSK3ARPS6KA3MAPK14
2'-Beta-Methyl-Guanosine SCHEMBL11965261 0.90 HINT1 (0.75) HINT1NT5EGSK3ARPS6KA3MAPK14
2'-Beta-Methyl-Guanosine SCHEMBL116165 0.90 HINT1 (0.75) HINT1NT5EGSK3ARPS6KA3MAPK14
SCHEMBL7111080 0.90 HINT1 (0.72) HINT1NT5EGSK3ARPS6KA3MAPK14
2'-Beta-Methyl-Guanosine SCHEMBL383785 0.90 HINT1 (0.75) HINT1NT5EGSK3ARPS6KA3MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002062924-A1 INSTANT DEGRADATION OF PLASTICS TO SOLUBLE NON-TOXIC PRODUCTS ROSEN OREN (IL) 2002-08-15 WO claimed
US-20020004590-A1 Method for producing nucleoside-5'-phosphate ester MIHARA YASUHIRO (JP) 2002-01-10 US claimed
US-5420105-A Drug delivery to targeted cells ALETHEON PHARMACEUTICALS, INC. 1995-05-30 US claimed
WO-2018231990-A2 POLYNUCLEOTIDES ENCODING METHYLMALONYL-COA MUTASE MODERNATX, INC. (US) 2018-12-20 WO disclosed
WO-2011069587-A1 LYOPHILIZATION OF NUCLEIC ACIDS IN LACTATE-CONTAINING SOLUTIONS CUREVAC GMBH (DE) 2011-06-16 WO disclosed
US-7575901-B2 Propagating escherichia mutant which produces 5'-inosinic acid or 5'-guanylic acid; identifying nucleotidase gene associated with generating nucleoside 5'-phosphate esters AJINOMOTO CO., INC. (JP) 2009-08-18 US disclosed
US-20080026428-A1 METHOD FOR PRODUCING NUCLEOTIDE BY FERMENTATION AJINOMOTO CO., INC. (JP) 2008-01-31 US disclosed
EP-0832970-B1 PROCESS FOR PRODUCING NUCLEOSIDE-5'-PHOSPHATE ESTER AJINOMOTO KK (JP) 2007-01-17 EP disclosed
EP-1170370-B1 Method for producing nucleotide by fermentation AJINOMOTO KK (JP) 2006-09-27 EP disclosed
US-20040152171-A1 Method for producing nucleotide by fermentation AJINOMOTO CO., INC. (JP) 2004-08-05 US disclosed
EP-0857788-B1 Method for producing nucleoside-5'-phosphate ester AJINOMOTO KK (JP) 2003-04-23 EP disclosed
WO-2002002172-A9 DNA PALINDROME - OLIGOGUANYLIC ACID COMPOSITIONS AND USES THEREOF UNIV JEFFERSON (US) 2002-07-18 WO disclosed
US-6355472-B2 ACID PHOSPHATASE AJINOMOTO CO., INC. (JP) 2002-03-12 US disclosed
US-20020004590-A1 Method for producing nucleoside-5'-phosphate ester MIHARA YASUHIRO (JP) 2002-01-10 US disclosed
EP-1170370-A2 Method for producing nucleotide by fermentation Ajinomoto Co., Inc. (JP) 2002-01-09 EP disclosed
US-6207435-B1 MUTANT ACID PHOSPHATASE HAVING DECREASED MICHAELIS CONSTANT FOR A NUCLEOSIDE AND/OR INCREASED TEMPERATURE STABILITY; FOR EFFICIENT PHOSPHORYLATION OF NUCLEOSIDES TO PRODUCE NUCLEOTIDES AJINOMOTO CO., INC. (JP) 2001-03-27 US disclosed
US-6015697-A ECONOMICAL AND EFFICIENT PROCESS BY REACTING A NUCLEOSIDE WITH A PHOSPHATE DONOR GROUP IN PRESENCE OF MUTANT ACID PHOSPHATASE WITH DECREASED MICHAELIS CONSTANT FOR NUCLEOSIDE OR INCREASED TEMPERATURE STABILITY AJINOMOTO CO., INC. (JP) 2000-01-18 US disclosed
US-6010851-A ALLOWING AN ACID PHOSPHATASE HAVING A LOWERED PHOSPHOMONOESTERASE ACTIVITY TO ACT UNDER A CONDITION OF PH 3.0 TO 5.5 ON A NUCLEOSIDE AND A PHOSPHATE GROUP DONOR AJINOMOTO CO., INC. (JP) 2000-01-04 US disclosed
EP-0857788-A2 Method for producing nucleoside-5'-phosphate ester Ajinomoto Co., Inc. (JP) 1998-08-12 EP disclosed
EP-0832970-A1 PROCESS FOR PRODUCING NUCLEOSIDE-5'-PHOSPHATE Ajinomoto Co., Inc. (JP) 1998-04-01 EP disclosed