SCHEMBL20141026

SCHEMBL20141026

COC(=O)c1cc(N(c2ccccc2OC(F)F)C2CCNCC2)c(C)cc1C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.41
SLC6A2 P23975 6/20 0.34
SLC6A4 P31645 6/20 0.34
DDB1 Q16531 1/20 0.34
CRBN Q96SW2 1/20 0.34
CCR8 P51685 1/20 0.33
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
KCNH2 Q12809 2/20 0.33
HPGD P15428 2/20 0.32
DVL1 O14640 1/20 0.32
DVL3 Q92997 1/20 0.32
CYP2D6 P10635 1/20 0.32
MTOR P42345 1/20 0.32
RPTOR Q8N122 1/20 0.32
MLST8 Q9BVC4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20140980 0.90 SLC6A2 (0.36) NR1I2SLC6A2SLC6A4KCNH2CYP2D6
SCHEMBL20141613 0.89 SLC6A2 (0.38) SLC6A2SLC6A4DDB1CRBNCCR8
SCHEMBL20140900 0.86 SLC6A2 (0.41) SLC6A2SLC6A4DDB1CRBN
SCHEMBL20141029 0.82 SLC6A2 (0.38) SLC6A2SLC6A4KCNH2HPGDDVL1
SCHEMBL20141738 0.80 SLC6A2 (0.40) SLC6A2SLC6A4CCR8KCNH2HPGD
SCHEMBL20141030 0.78 SLC6A2 (0.38) SLC6A2SLC6A4HPGD
SCHEMBL20141036 0.77 KCNH2 (0.37) SLC6A2SLC6A4KCNH2HPGDCYP2D6
SCHEMBL20141038 0.77 KCNH2 (0.37) SLC6A2SLC6A4KCNH2HPGDCYP2D6
SCHEMBL20141346 0.77 SLC6A2 (0.44) SLC6A2SLC6A4KCNH2CYP2D6
SCHEMBL20141147 0.77 SLC6A2 (0.38) SLC6A2SLC6A4KCNH2HPGDDVL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538091-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF Navitor Pharmaceuticals, Inc. (US) 2019-09-18 EP disclosed
WO-2018089499-A1 PHENYL AMINO PIPERIDINE mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed