SCHEMBL2014124

SCHEMBL2014124

Cc1nn2c(C(=O)N(C)C(CCNC(=O)c3cccn3C)Cc3ccccc3)cnc2s1

nearest known ligand 0.59

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.59
HCRTR2 O43614 2/20 0.59
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
HDAC6 Q9UBN7 3/20 0.38
HRH3 Q9Y5N1 2/20 0.37
PADI4 Q9UM07 3/20 0.36
IDO1 P14902 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013002 0.87 HCRTR1 (0.57) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL2013001 0.86 HCRTR1 (0.56) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL6918074 0.84 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL2014627 0.84 HCRTR1 (0.59) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL2015686 0.84 HCRTR1 (0.55) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL2014249 0.82 HCRTR1 (0.61) HCRTR1HCRTR2NPC1RAB9AHRH3
SCHEMBL13139060 0.81 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL2051297 0.80 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL2012749 0.80 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AHDAC6
SCHEMBL2014992 0.80 HCRTR1 (0.62) HCRTR1HCRTR2NPC1RAB9AHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO claimed
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed