SCHEMBL20141840

SCHEMBL20141840

Cc1ccc(CN2CCN(c3ncccc3C#N)CC2)cc1C(=O)N1CCN(c2ccccc2C#N)C[C@@H]1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 3/20 0.49
PARP1 P09874 2/20 0.45
TNK2 Q07912 1/20 0.45
TNK1 Q13470 1/20 0.45
DRD2 P14416 4/20 0.44
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HTR2A P28223 3/20 0.43
HTR1A P08908 1/20 0.43
HTR7 P34969 1/20 0.43
MTOR P42345 2/20 0.42
RPTOR Q8N122 2/20 0.42
MLST8 Q9BVC4 2/20 0.42
DRD4 P21917 2/20 0.42
CHRM4 P08173 1/20 0.42
HSD11B1 P28845 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CHRM2 P08172 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20156810 0.94 MTOR (0.47) GRM1PARP1TNK2TNK1DRD2
SCHEMBL20157309 0.94 MTOR (0.47) GRM1PARP1TNK2TNK1DRD2
SCHEMBL20142175 0.91 GRM1 (0.50) GRM1DRD2KDM4EALDH1A1HTR2A
SCHEMBL20157005 0.89 CHRM4 (0.47) GRM1KDM4EALDH1A1MTORRPTOR
SCHEMBL20157004 0.89 CHRM4 (0.47) GRM1KDM4EALDH1A1MTORRPTOR
SCHEMBL20140106 0.88 GRM1 (0.47) GRM1PARP1TNK2TNK1KDM4E
SCHEMBL20157186 0.87 MTOR (0.55) GRM1DRD2KDM4EALDH1A1MTOR
SCHEMBL20157188 0.87 MTOR (0.55) GRM1DRD2KDM4EALDH1A1MTOR
SCHEMBL20140600 0.87 KDM4E (0.54) PARP1TNK2TNK1DRD2KDM4E
SCHEMBL20157075 0.86 CHRM4 (0.49) GRM1MTORRPTORMLST8CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed
WO-2018089433-A1 PHENYL mTORC INHIBITORS AND USES THEREOF NAVITOR PHARMACEUTICALS, INC. (US) 2018-05-17 WO disclosed