SCHEMBL20142267

SCHEMBL20142267

Cc1ccc(Nc2nc(N(C)C)c(C(=O)c3ccncc3)s2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.51
GSK3B P49841 2/20 0.51
CDK5 Q00535 8/20 0.50
CDK5R1 Q15078 8/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ADORA3 P0DMS8 4/20 0.49
ADORA2A P29274 3/20 0.49
ADORA1 P30542 3/20 0.49
NPC1 O15118 5/20 0.49
RAB9A P51151 4/20 0.49
MAPT P10636 3/20 0.49
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
MAPK14 Q16539 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ADORA2B P29275 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20142841 0.89 MAPT (0.63) GSK3AGSK3BCDK5CDK5R1SMN1; SMN2
SCHEMBL20142501 0.87 CDK5 (0.49) GSK3AGSK3BCDK5CDK5R1ADORA3
SCHEMBL20142409 0.87 GSK3A (0.53) GSK3AGSK3BCDK5CDK5R1SMN1; SMN2
SCHEMBL20142179 0.87 GSK3A (0.53) GSK3AGSK3BCDK5CDK5R1SMN1; SMN2
SCHEMBL20142075 0.86 CCNA2 (0.59) GSK3AGSK3BCDK5CDK5R1SMN1; SMN2
SCHEMBL20142448 0.84 GSK3A (0.73) GSK3AGSK3BCDK5CDK5R1SMN1; SMN2
SCHEMBL20142465 0.84 CDK5 (0.52) CDK5CDK5R1SMN1; SMN2ADORA3ADORA2A
SCHEMBL20142417 0.83 CCNA2 (0.57) GSK3AGSK3BCDK5CDK5R1SMN1; SMN2
SCHEMBL20142455 0.83 GSK3A (0.71) GSK3AGSK3BCDK5CDK5R1NPC1
SCHEMBL20142420 0.81 CDK5 (0.51) GSK3AGSK3BCDK5CDK5R1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO claimed
WO-2018089902-A1 DIAMINOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE APOGEE BIOTECHNOLOGY CORPORATION (US) 2018-05-17 WO disclosed