SCHEMBL20142649

SCHEMBL20142649

Nc1ccnc(N2CCCC2)c1N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
TSHR P16473 3/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 2/20 0.45
GLA P06280 1/20 0.45
LMNA P02545 1/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MAPT P10636 2/20 0.42
NUDT1 P36639 1/20 0.42
HTT P42858 1/20 0.40
MAPK1 P28482 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
GFER P55789 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HPGD P15428 1/20 0.39
JAK3 P52333 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30281019 1.00 KDM4E (0.45) KDM4ETSHRALDH1A1GAAGLA
SCHEMBL17555901 0.98 ALDH1A1 (0.47) KDM4ETSHRALDH1A1GAAGLA
SCHEMBL17555848 0.83 HRH4 (0.53) KDM4EALDH1A1GAAMAPTGFER
SCHEMBL8745499 0.83 HTR2C (0.53)
SCHEMBL30622679 0.83 KDM4E (0.57) KDM4EALDH1A1GAALMNACYP1A2
SCHEMBL17583342 0.83 KDM4E (0.57) KDM4EALDH1A1GAALMNACYP1A2
SCHEMBL17583291 0.82 SCN10A (0.40) HTT
SCHEMBL3947341 0.77 ALDH1A1 (0.45) KDM4ETSHRALDH1A1GAAGLA
SCHEMBL2899027 0.77 DYRK1A (0.46) KDM4ETSHRALDH1A1GAAGLA
SCHEMBL29508931 0.76 GRIN2D (0.58) KDM4ETSHRALDH1A1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538088-A1 HETEROCYCLIC MODULATORS OF LIPID SYNTHESIS 3-V Biosciences, Inc. (US) 2019-09-18 EP disclosed
WO-2018089904-A1 HETEROCYCLIC MODULATORS OF LIPID SYNTHESIS 3-V BIOSCIENCES, INC. (US) 2018-05-17 WO disclosed