SCHEMBL20142949

SCHEMBL20142949

CC(CC(=O)c1ccc(Br)cc1)(C(=O)O)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.52
HDAC1 Q13547 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
HDAC9 Q9UKV0 1/20 0.48
HDAC5 Q9UQL6 1/20 0.48
HAO1 Q9UJM8 1/20 0.46
NPC1 O15118 2/20 0.44
HPGD P15428 2/20 0.44
RAB9A P51151 2/20 0.44
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
KMT2A Q03164 4/20 0.41
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL180665 0.87 GSK3B (0.53) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL8531622 0.82 MAPT (0.52) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL10021821 0.82 GSK3B (0.57) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL28303452 0.82 GSK3B (0.48) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL20530433 0.81 GSK3B (0.50) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL8534141 0.80 MAPT (0.59) GSK3BHAO1NPC1HPGDRAB9A
SCHEMBL20159373 0.80 ALDH1A1 (0.50) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL1748168 0.76 GSK3B (0.46) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL1748024 0.75 GSK3B (0.48) GSK3BHDAC1HDAC8HDAC3HDAC4
SCHEMBL10645626 0.75 HDAC1 (0.42) GSK3BHDAC1HDAC8HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed