SCHEMBL20143637

SCHEMBL20143637

CC(C)(C)OC(=O)N1Cc2cc(C(=O)OCc3ccccc3)ccc2C[C@@H]1C(=O)OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 5/20 0.50
HDAC8 Q9BY41 9/20 0.49
NPSR1 Q6W5P4 1/20 0.45
ACE P12821 1/20 0.43
GPR119 Q8TDV5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17486403 0.92 PTPN1 (0.50) PTPN1HDAC8NPSR1ACE
SCHEMBL8233145 0.88 NPSR1 (0.53) PTPN1HDAC8NPSR1
SCHEMBL29727828 0.88 NPSR1 (0.53) PTPN1HDAC8NPSR1
SCHEMBL7228636 0.84 ACE (0.59) PTPN1HDAC8NPSR1ACE
SCHEMBL7228628 0.84 ACE (0.59) PTPN1HDAC8NPSR1ACE
SCHEMBL3615808 0.81 HDAC8 (0.49) PTPN1HDAC8NPSR1ACE
SCHEMBL31162867 0.81 NR1H2 (0.57) GPR119
SCHEMBL6787776 0.80 FKBP1A (0.49) PTPN1
SCHEMBL204506 0.80 FKBP1A (0.49) PTPN1
SCHEMBL204505 0.80 FKBP1A (0.49) PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9969709-B2 Guanidinobenzoic acid ester compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-05-15 US disclosed