SCHEMBL20143674

SCHEMBL20143674

CCOC(=O)C(C)(C)CC(=O)c1ccc(Br)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
MAPT P10636 5/20 0.50
KMT2A Q03164 4/20 0.50
HPGD P15428 2/20 0.50
NPSR1 Q6W5P4 3/20 0.48
POLB P06746 1/20 0.48
LMNA P02545 3/20 0.46
GSK3B P49841 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC11 Q96DB2 1/20 0.43
HDAC8 Q9BY41 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20159373 0.90 ALDH1A1 (0.50) ALDH1A1MAPTKMT2AHPGDNPSR1
SCHEMBL1373141 0.85 ESR1 (0.56) ALDH1A1MAPTNPSR1POLBNPC1
SCHEMBL10596544 0.84 TSHR (0.56) ALDH1A1MAPTKMT2AHPGDNPSR1
SCHEMBL12121920 0.83 POLB (0.66) ALDH1A1MAPTKMT2AHPGDNPSR1
SCHEMBL1748024 0.83 GSK3B (0.48) ALDH1A1MAPTKMT2AHPGDNPSR1
SCHEMBL1747922 0.82 ALDH1A1 (0.51) ALDH1A1MAPTKMT2AHPGDNPSR1
SCHEMBL4232023 0.80 LMNA (0.53) ALDH1A1MAPTKMT2AHPGDNPSR1
SCHEMBL12912525 0.80 ALDH1A1 (0.52) ALDH1A1MAPTKMT2AHPGDNPSR1
SCHEMBL21294046 0.79 ALDH1A1 (0.44) ALDH1A1MAPTKMT2ANPSR1POLB
SCHEMBL7799487 0.79 ALDH1A1 (0.49) ALDH1A1MAPTKMT2AHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021013693-A1 ANTIBODY DRUG CONJUGATES (ADCS) WITH NAMPT INHIBITORS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2021-01-28 WO disclosed
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed
WO-2018086703-A1 DIHYDROPYRIDAZINONES SUBSTITUTED WITH PHENYLUREAS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-17 WO disclosed