SCHEMBL20144317

SCHEMBL20144317

Cc1ccc(-c2nc3ccc(CN4CCN(C)CC4)cc3[nH]2)cc1C#C/C(N)=C/C=C(\N)NC1CCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.44
HDAC3 O15379 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
GSK3B P49841 2/20 0.43
FGFR1 P11362 6/20 0.41
FLT1 P17948 2/20 0.41
AURKA O14965 3/20 0.40
AURKB Q96GD4 3/20 0.40
CDK1 P06493 2/20 0.40
CCNB1 P14635 2/20 0.40
CDK2 P24941 1/20 0.40
KDR P35968 4/20 0.39
PDGFRB P09619 1/20 0.39
FGFR2 P21802 4/20 0.39
FGFR3 P22607 4/20 0.39
KIT P10721 4/20 0.38
BMPR1B O00238 1/20 0.38
CDC7 O00311 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20144320 0.97 HDAC3 (0.45) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL20144350 0.92 HDAC6 (0.45) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL20144335 0.89 HDAC3 (0.46) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL20144361 0.89 HDAC6 (0.46) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL20144341 0.81 HDAC6 (0.47) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL15443033 0.78 HDAC6 (0.44) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL15442177 0.75 ABL1 (0.48) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL15442319 0.74 HDAC3 (0.45) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL15442505 0.74 HDAC6 (0.46) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL15442512 0.71 FGFR1 (0.57) HDAC6HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3186247-B1 PROTEIN KINASE INHIBITORS ASTAR BIOTECH LLC (US) 2021-03-03 EP disclosed
EP-2880038-B1 PROTEIN KINASE INHIBITORS ASTAR BIOTECH LLC (US) 2018-05-16 EP disclosed