SCHEMBL20144462

SCHEMBL20144462

COC(=O)/C(SN1CCOCC1)=C(/C)N

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RECQL P46063 1/20 0.40
GLA P06280 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 2/20 0.33
BLM P54132 1/20 0.33
MGLL Q99685 2/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
TSHR P16473 2/20 0.31
HTT P42858 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19525077 0.81 RECQL (0.35) RECQLGLASMN1; SMN2ALDH1A1KDM4E
SCHEMBL5175953 0.70 MGLL (0.46) GLASMN1; SMN2ALDH1A1KDM4EMGLL
SCHEMBL29194966 0.66 MGLL (0.41) RECQLGLASMN1; SMN2ALDH1A1MGLL
SCHEMBL11044755 0.66 MGLL (0.50) GLASMN1; SMN2ALDH1A1KDM4EMGLL
SCHEMBL10560780 0.64 MGLL (0.48) GLASMN1; SMN2ALDH1A1KDM4EMGLL
SCHEMBL30709623 0.64 MGLL (0.48) GLASMN1; SMN2ALDH1A1KDM4EMGLL
SCHEMBL23673842 0.64 ALDH1A1 (0.52) RECQLGLASMN1; SMN2ALDH1A1BLM
SCHEMBL27924627 0.63 MGLL (0.46) ALDH1A1KDM4EMGLLHPGD
SCHEMBL29141222 0.63 MGLL (0.46) SMN1; SMN2ALDH1A1MGLL
SCHEMBL3452606 0.62 MGLL (0.41) SMN1; SMN2ALDH1A1KDM4EMGLLHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3321257-A1 SUBSTITUTED 5-AMINOTHIENO[2,3-C]PYRIDAZINE-6-CARBOXAMIDE ANALOGS AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 Vanderbilt University (US) 2018-05-16 EP disclosed