SCHEMBL20144682

SCHEMBL20144682

COC(=O)[C@H](C/C=C/C1CCCC1)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 0.44
NFKB2 Q00653 2/20 0.44
RELA Q04206 2/20 0.44
CTSK P43235 6/20 0.43
CTSS P25774 2/20 0.43
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
CACNA1B Q00975 6/20 0.41
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
AAK1 Q2M2I8 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
CTSL P07711 1/20 0.36
EPHX1 P07099 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL375737 0.88 CTSK (0.46) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL25139692 0.88 CTSK (0.46) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL29178408 0.86 CTSK (0.45) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL30047908 0.86 CTSK (0.45) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL17884307 0.83 CTSK (0.54) NFKB1NFKB2RELACTSKCTSS
SCHEMBL16330414 0.83 CTSK (0.54) NFKB1NFKB2RELACTSKCTSS
SCHEMBL6885122 0.81 HDAC4 (0.41) NFKB1NFKB2RELACTSKCTSS
SCHEMBL28690504 0.80 CTSK (0.48) NFKB1NFKB2RELACTSKCTSS
SCHEMBL28690502 0.80 CTSK (0.48) NFKB1NFKB2RELACTSKCTSS
SCHEMBL17880416 0.78 CTSK (0.49) NFKB1NFKB2RELACTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2751124-B1 VERSATILE AND STEREOSPECIFIC SYNTHESIS OF GAMMA,DELTA -UNSATURATED AMINO ACIDS BY WITTIG REACTION CENTRE NAT RECH SCIENT (FR) 2018-05-16 EP disclosed