SCHEMBL29178408

SCHEMBL29178408

CNC(=O)C(CC=CC1CCCC1)NC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.45
CTSS P25774 6/20 0.45
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
CACNA1B Q00975 4/20 0.39
AAK1 Q2M2I8 2/20 0.37
CTSL P07711 2/20 0.36
CTSB P07858 1/20 0.36
KMT2A Q03164 1/20 0.36
EPHX1 P07099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30047908 1.00 CTSK (0.45) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL25139692 0.87 CTSK (0.46) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL375737 0.87 CTSK (0.46) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL20144682 0.86 NFKB1 (0.44) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL29178395 0.79 CTSK (0.48) CTSKCTSSCTSLCTSB
SCHEMBL29178398 0.79 CTSK (0.48) CTSKCTSSCTSLCTSB
SCHEMBL24815288 0.79 CTSK (0.48) CTSKCTSSCTSLCTSB
SCHEMBL24812376 0.76 CTSK (0.44) CTSKCTSSCTSLCTSB
SCHEMBL29178308 0.76 CTSK (0.44) CTSKCTSSCTSLCTSB
SCHEMBL25139652 0.74 HDAC4 (0.56) CTSKCTSSHDAC4HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117561058-A CDK2 inhibitors and methods of use thereof 塞迪拉治疗股份有限公司 2024-02-13 CN disclosed