SCHEMBL20144784

SCHEMBL20144784

CCOc1ccccc1C(=O)N1CCCC(Nc2ccc(C(F)(F)F)cn2)C1

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 10/20 0.69
HCRTR1 O43613 9/20 0.69
SMN1; SMN2 Q16637 3/20 0.62
KDM4E B2RXH2 2/20 0.62
LMNA P02545 1/20 0.62
ALDH1A1 P00352 1/20 0.51
HTT P42858 1/20 0.51
MAP3K12 Q12852 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18697642 1.00 HCRTR2 (0.69) HCRTR2HCRTR1SMN1; SMN2KDM4ELMNA
SCHEMBL20144919 0.86 HCRTR2 (0.67) HCRTR2HCRTR1SMN1; SMN2KDM4ELMNA
SCHEMBL20145234 0.86 HCRTR2 (0.67) HCRTR2HCRTR1SMN1; SMN2KDM4ELMNA
SCHEMBL20145031 0.83 HCRTR2 (0.70) HCRTR2HCRTR1
SCHEMBL20144824 0.83 HCRTR2 (0.70) HCRTR2HCRTR1
SCHEMBL20144897 0.82 HCRTR2 (0.68) HCRTR2HCRTR1LMNA
SCHEMBL18697634 0.81 HCRTR2 (0.69) HCRTR2HCRTR1
SCHEMBL20144748 0.81 HCRTR2 (0.69) HCRTR2HCRTR1
SCHEMBL16031595 0.81 HCRTR1 (1.00) HCRTR2HCRTR1
SCHEMBL16030577 0.81 HCRTR1 (1.00) HCRTR2HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed