SCHEMBL20144917

SCHEMBL20144917

COc1ccc(C(=O)N2CCCC(Nc3ncc(Cl)cn3)C2)c(-n2nccn2)c1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 14/20 0.56
HCRTR2 O43614 13/20 0.54
GAA P10253 1/20 0.50
CCNK O75909 3/20 0.48
CDK12 Q9NYV4 3/20 0.48
GFER P55789 1/20 0.48
CCNA2 P20248 2/20 0.48
CDK2 P24941 2/20 0.48
CDK7 P50613 2/20 0.48
CCNH P51946 2/20 0.48
MNAT1 P51948 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18697732 1.00 HCRTR1 (0.56) HCRTR1HCRTR2GAACCNKCDK12
SCHEMBL18697651 0.91 HCRTR1 (0.55) HCRTR1HCRTR2GAAGFER
SCHEMBL20144971 0.91 HCRTR1 (0.55) HCRTR1HCRTR2GAAGFER
SCHEMBL20144834 0.89 HCRTR1 (0.71) HCRTR1HCRTR2GAA
SCHEMBL20144988 0.89 HCRTR1 (0.68) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL18697535 0.89 HCRTR1 (0.68) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL20145000 0.86 HCRTR1 (0.55) HCRTR1HCRTR2GAACCNKCDK12
SCHEMBL20144741 0.85 HCRTR2 (0.65) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20144731 0.82 HCRTR1 (0.71) HCRTR1HCRTR2GFER
SCHEMBL16148077 0.82 HCRTR1 (0.81) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed