SCHEMBL20144988

SCHEMBL20144988

Cc1ccc(C(=O)N2CCCC(Nc3ncc(Cl)cn3)C2)c(-n2nccn2)c1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 15/20 0.68
HCRTR2 O43614 9/20 0.68
CCNK O75909 2/20 0.52
CDK12 Q9NYV4 2/20 0.52
GFER P55789 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18697535 1.00 HCRTR1 (0.68) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL18697656 0.90 HCRTR1 (0.69) HCRTR1HCRTR2GFER
SCHEMBL20144828 0.90 HCRTR1 (0.69) HCRTR1HCRTR2GFER
SCHEMBL20144917 0.89 HCRTR1 (0.56) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL20144982 0.89 HCRTR1 (0.70) HCRTR1HCRTR2
SCHEMBL18697732 0.89 HCRTR1 (0.56) HCRTR1HCRTR2CCNKCDK12GFER
SCHEMBL20144741 0.87 HCRTR2 (0.65) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20145124 0.86 HCRTR1 (0.68) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20144928 0.86 HCRTR1 (0.68) HCRTR1HCRTR2CCNKCDK12
SCHEMBL20145252 0.86 HCRTR1 (0.69) HCRTR1HCRTR2CCNKCDK12GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed