SCHEMBL20145208

SCHEMBL20145208

O=CN1CCCC(Nc2ccc(C(F)(F)F)cn2)C1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR6 P51684 5/20 0.51
DPP4 P27487 2/20 0.49
HCRTR1 O43613 7/20 0.46
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
CYP2C9 P11712 2/20 0.45
HSD11B1 P28845 2/20 0.45
CCNK O75909 1/20 0.45
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CDK12 Q9NYV4 1/20 0.45
HCRTR2 O43614 3/20 0.44
TRPV1 Q8NER1 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20144869 0.82 IL1B (0.55) CCR6DPP4CCNKCCNA2CDK2
SCHEMBL20145261 0.82 IL1B (0.55) CCR6DPP4CCNKCCNA2CDK2
SCHEMBL20145167 0.81 CCNK (0.48) CCR6DPP4HCRTR1CCNKCDK12
SCHEMBL31308025 0.81 CCR6 (0.51) CCR6DPP4HCRTR1CCNKCCNA2
SCHEMBL15739705 0.80 HCRTR1 (0.55) CCR6DPP4HCRTR1CCNKCCNA2
SCHEMBL18607634 0.80 CCR6 (0.55) CCR6DPP4HCRTR1CCNKCCNA2
SCHEMBL30955917 0.77 CCNK (0.47) CCR6HCRTR1CCNKCDK2CDK12
SCHEMBL15739645 0.77 CCR6 (0.61) CCR6DPP4HCRTR1
SCHEMBL16032596 0.75 HCRTR1 (0.59) HCRTR1HCRTR2
SCHEMBL16730436 0.74 CCR6 (0.58) CCR6DPP4CCNKCCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed