SCHEMBL20145167

SCHEMBL20145167

O=CN1CCCC(Nc2ccc(Cl)cn2)C1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCNK O75909 2/20 0.48
CDK12 Q9NYV4 2/20 0.48
DPP4 P27487 1/20 0.45
LMNA P02545 3/20 0.45
GAA P10253 2/20 0.45
TSHR P16473 2/20 0.44
HCAR3 P49019 2/20 0.42
HCRTR1 O43613 3/20 0.41
HCRTR2 O43614 2/20 0.41
GRM5 P41594 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CCR6 P51684 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KDM4E B2RXH2 1/20 0.40
USP30 Q70CQ3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20145228 0.81 IL1B (0.54) CCNKCDK12
SCHEMBL20145208 0.81 CCR6 (0.51) CCNKCDK12DPP4HCRTR1HCRTR2
SCHEMBL28545513 0.75 MAPK1 (0.49) CCNKCDK12
SCHEMBL28545510 0.75 MAPK1 (0.49) CCNKCDK12
SCHEMBL28552999 0.75 CCNK (0.60) CCNKCDK12LMNAGAAHCAR3
SCHEMBL28552998 0.75 CCNK (0.60) CCNKCDK12LMNAGAAHCAR3
SCHEMBL15739537 0.75 HCAR3 (0.56) CCNKCDK12TSHRHCAR3L3MBTL1
SCHEMBL23073961 0.74 HSD11B1 (0.39) DPP4LMNAGAATSHR
SCHEMBL13592662 0.74 HSD11B1 (0.39) DPP4LMNAGAATSHR
Hydrochloric Acid SCHEMBL28911922 0.74 MAPK1 (0.48) CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed