SCHEMBL20145226

SCHEMBL20145226

Brc1ccc(OC2CCCNC2)nc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.49
CHRNA4 P43681 4/20 0.49
ROCK1 Q13464 5/20 0.45
ROCK2 O75116 3/20 0.44
KCNH2 Q12809 1/20 0.44
MKNK1 Q9BUB5 2/20 0.43
CDC42BPB Q9Y5S2 2/20 0.40
CDC42BPA Q5VT25 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40
DGAT1 O75907 1/20 0.39
IKBKB O14920 1/20 0.39
CHUK O15111 1/20 0.39
HTR1A P08908 1/20 0.39
SLC6A2 P23975 1/20 0.39
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
PIM1 P11309 1/20 0.38
PIM2 Q9P1W9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4828298 0.91 CHRNB2 (0.47) CHRNB2CHRNA4MKNK1DGAT1
SCHEMBL10078051 0.84 SLC6A4 (0.43) DGAT1
SCHEMBL30314525 0.84 SLC6A4 (0.43) DGAT1
Hydrochloric Acid SCHEMBL517567 0.83 SLC6A4 (0.42) DGAT1
Hydrochloric Acid SCHEMBL31347800 0.83 SLC6A4 (0.42) DGAT1
SCHEMBL1928105 0.82 DGAT1 (0.47) KCNH2DGAT1
SCHEMBL4000064 0.82 DGAT1 (0.47) KCNH2DGAT1
SCHEMBL30296157 0.82 DGAT1 (0.47) KCNH2DGAT1
SCHEMBL28671509 0.82 CHRNB2 (0.49) CHRNB2CHRNA4ROCK1ROCK2KCNH2
SCHEMBL29517983 0.82 CHRNB2 (0.49) CHRNB2CHRNA4ROCK1ROCK2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed