SCHEMBL2014680

SCHEMBL2014680

C[C@H](N)C(=O)Oc1ccccc1F

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
GAA P10253 1/20 0.51
CARM1 Q86X55 2/20 0.47
PRMT6 Q96LA8 2/20 0.47
LMNA P02545 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.43
PARP10 Q53GL7 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
FAAH O00519 4/20 0.41
KMT2A Q03164 2/20 0.41
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
TP53 P04637 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CXCL8 P10145 1/20 0.39
MEN1 O00255 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15670768 1.00 ALDH1A1 (0.51) ALDH1A1GAACARM1PRMT6LMNA
SCHEMBL17260382 0.86 ALDH1A1 (0.42) ALDH1A1GAACARM1PRMT6LMNA
SCHEMBL4596733 0.85 ALDH1A1 (0.50) ALDH1A1GAALMNASMN1; SMN2MAPT
SCHEMBL1822201 0.84 ALDH1A1 (0.49) ALDH1A1GAALMNASMN1; SMN2MAPT
SCHEMBL28063973 0.83 L3MBTL1 (0.46) ALDH1A1CARM1PRMT6LMNAMAPT
SCHEMBL27945186 0.83 CYP4F2 (0.41) ALDH1A1GAACARM1PRMT6
SCHEMBL8791825 0.82 ALDH1A1 (0.47) ALDH1A1GAALMNASMN1; SMN2MAPT
SCHEMBL21635123 0.81 ALDH1A1 (0.55) ALDH1A1GAACARM1PRMT6LMNA
SCHEMBL1983875 0.80 TSHR (0.46) ALDH1A1GAASMN1; SMN2MAPTHPGD
SCHEMBL935390 0.80 KMT2A (0.43) ALDH1A1GAACARM1PRMT6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1112125-A Acyloxyhexanoic acid derivatives CIBA GEIGY AG (CH) 1995-11-22 CN claimed
JP-3160985-A None JP disclosed
JP-6189694-A None JP disclosed
WO-2025262025-A1 PHARMACEUTICAL COMPOSITION FOR PASSIVE IMMUNIZATION OR THERAPY HEIDELBERG BIOTECH GMBH (DE) 2025-12-26 WO disclosed
WO-2025262082-A1 UNIVERSAL PRINCIPLES OF ACTIVE AND PASSIVE IMMUNIZATION AGAINST VIRAL ANTIGENS HEIDELBERG BIOTECH GMBH (DE) 2025-12-26 WO disclosed
WO-2025262023-A1 PROTEIN OLIGOMERS FOR ACTIVE IMMUNIZATION HEIDELBERG BIOTECH GMBH (DE) 2025-12-26 WO disclosed
US-12428455-B2 Dominant negative CEBPB and CEBPD proteins and methods of use for decreasing viability of neoplastic cells THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2025-09-30 US disclosed
US-20250223328-A1 TRUNCATED DOMINANT NEGATIVE CEBPB AND CEBPD PROTEINS AND METHODS OF USE FOR DECREASING VIABILITY OF NEOPLASTIC CELLS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2025-07-10 US disclosed
CN-113396218-B Engineered transaminase polypeptides 科德克希思公司 2025-02-18 CN disclosed
EP-4358989-A2 BICYCLIC PEPTIDYL PAN-RAS INHIBITORS Ohio State Innovation Foundation (US) 2024-05-01 EP disclosed
EP-0663897-B1 PROCESS FOR SEPARATING ENANTIOMERS FROM A RACEMIC MIXTURE AKZO NOBEL NV (NL) 1997-01-29 EP disclosed
US-5514773-A PARASITICIDES, ANTHELMINTICS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-05-07 US disclosed
WO-1996011894-A1 PROCESS FOR SEPARATING ENANTIOMERS FROM A RACEMIC MIXTURE AKZO NOBEL N.V. (NL) 1996-04-25 WO disclosed
CN-1112125-A Acyloxyhexanoic acid derivatives CIBA GEIGY AG (CH) 1995-11-22 CN disclosed
EP-0663897-A1 PROCESS FOR SEPARATING ENANTIOMERS FROM A RACEMIC MIXTURE. AKZO NOBEL NV (NL) 1995-07-26 EP disclosed
EP-0634408-A1 DEPSIPEPTIDE DERIVATIVE, PRODUCTION THEREOF AND USE THEREOF FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-01-18 EP disclosed
JP-H06189694-A PRODUCTION OF FOOD AND DRINK KYOWA HAKKO KOGYO CO LTD 1994-07-12 JP disclosed
WO-1994007814-A1 PROCESS FOR SEPARATING ENANTIOMERS FROM A RACEMIC MIXTURE AKZO NOBEL N.V. (NL) 1994-04-14 WO disclosed
JP-H03160985-A NOVEL VARIANT AND PREPARATION OF SOY SAUCE USING THEREOF KIKKOMAN CORP 1991-07-10 JP disclosed
EP-0331404-A2 Method for producing tropane alkaloid SEITAIKINOU RIYOU KAGAKUHIN SHINSEIZOUGIJUTSU KENKYU KUMIAI (JP) 1989-09-06 EP disclosed