SCHEMBL2014766

SCHEMBL2014766

O=C(NCc1cccnc1)C1CCC(c2ccccc2)N(S(=O)(=O)c2ccccc2)C1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.60
ALDH1A1 P00352 4/20 0.59
CYP2C9 P11712 3/20 0.56
CYP2C19 P33261 3/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
KMT2A Q03164 3/20 0.56
LMNA P02545 2/20 0.56
SMN1; SMN2 Q16637 1/20 0.56
MEN1 O00255 1/20 0.56
MAPK1 P28482 1/20 0.56
CYP1A2 P05177 1/20 0.52
NAMPT P43490 1/20 0.52
MAPT P10636 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12628516 1.00 TSHR (0.60) TSHRALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL2016227 0.94 ALDH1A1 (0.67) TSHRALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL12628517 0.94 ALDH1A1 (0.67) TSHRALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL12628161 0.90 ALDH1A1 (0.48) TSHRALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL2011504 0.90 ALDH1A1 (0.54) ALDH1A1KMT2AMEN1MAPT
SCHEMBL12628159 0.90 ALDH1A1 (0.54) ALDH1A1KMT2AMEN1MAPT
SCHEMBL12628514 0.89 ALDH1A1 (0.55) TSHRALDH1A1KMT2AMEN1MAPT
SCHEMBL2012792 0.89 ALDH1A1 (0.55) TSHRALDH1A1KMT2AMEN1MAPT
SCHEMBL12628168 0.85 KMT2A (0.52) TSHRALDH1A1CYP2C9CYP2C19CYP3A4
SCHEMBL2016260 0.85 KMT2A (0.52) TSHRALDH1A1CYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073269-A1 PIPERIDINE ARYL SULFONAMIDE DERIVATIVES AS KV1.3 MODULATORS EVOTEC AG (DE) 2011-06-23 WO claimed