SCHEMBL20149032

SCHEMBL20149032

CC(c1ccc([C@@H]2CN(C(=O)OCc3ccccc3)C[C@@H]2c2ccccc2)cc1)(C(F)(F)F)C(F)(F)F

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RORC P51449 8/20 0.58
PDK1 Q15118 1/20 0.48
PDK2 Q15119 1/20 0.48
PDK3 Q15120 1/20 0.48
PDK4 Q16654 1/20 0.48
KDM1A O60341 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HTT P42858 1/20 0.44
TACR1 P25103 2/20 0.44
TSHR P16473 1/20 0.44
PDE4B Q07343 2/20 0.44
HTR2C P28335 1/20 0.44
GPBAR1 Q8TDU6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20149087 0.78 RORC (0.75) RORC
SCHEMBL349184 0.77 SMN1; SMN2 (0.53) KDM1ANPC1RAB9ASMN1; SMN2HTT
SCHEMBL10683024 0.74 SMN1; SMN2 (0.57) KDM1ANPC1RAB9ASMN1; SMN2HTT
SCHEMBL10683021 0.74 SMN1; SMN2 (0.57) KDM1ANPC1RAB9ASMN1; SMN2HTT
SCHEMBL10683015 0.74 SMN1; SMN2 (0.57) KDM1ANPC1RAB9ASMN1; SMN2HTT
SCHEMBL16472054 0.74 SMN1; SMN2 (0.57) RORCPDK1PDK2PDK3PDK4
SCHEMBL16158890 0.74 SMN1; SMN2 (0.58) KDM1ANPC1RAB9ASMN1; SMN2HTT
SCHEMBL31412573 0.74 SMN1; SMN2 (0.47) KDM1ANPC1RAB9ASMN1; SMN2PDE4B
SCHEMBL20149112 0.74 RORC (1.00) RORCTACR1
SCHEMBL20149129 0.72 RORC (0.80) RORCTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed