SCHEMBL20149129

SCHEMBL20149129

CC(=O)N1CCC(C(=O)N2C[C@@H](c3ccccc3)[C@H](c3ccc(C(C)(C(F)(F)F)C(F)(F)F)cc3)C2)CC1

nearest known ligand 0.80

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RORC P51449 13/20 0.80
TACR1 P25103 7/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
NR1I2 O75469 2/20 0.54
TACR2 P21452 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23713056 0.89 RORC (1.00) RORCTACR1CYP3A4CYP2D6CYP2C9
SCHEMBL20149050 0.80 RORC (0.84) RORCTACR1NR1I2TACR2
SCHEMBL20149126 0.80 RORC (0.83) RORCNR1I2
SCHEMBL23713117 0.78 RORC (1.00) RORCTACR1CYP3A4CYP2D6CYP2C9
SCHEMBL20149032 0.72 RORC (0.58) RORCTACR1
SCHEMBL20149057 0.72 RORC (1.00) RORCTACR1NR1I2
SCHEMBL4144315 0.72 TACR1 (0.78) RORCTACR1CYP3A4CYP2D6CYP2C9
SCHEMBL4144312 0.72 TACR1 (0.78) RORCTACR1CYP3A4CYP2D6CYP2C9
SCHEMBL4483139 0.72 TACR1 (0.67) RORCTACR1CYP3A4CYP2D6CYP2C9
SCHEMBL4483149 0.72 TACR1 (0.67) RORCTACR1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089406-A1 ROR GAMMA MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed