SCHEMBL20150686

SCHEMBL20150686

C=CC(=O)Nc1cccc(Nc2ncnc3[nH]c(-c4ccc(NCCO)cc4)cc23)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.50
SRC P12931 5/20 0.50
FYN P06241 4/20 0.50
ERBB2 P04626 3/20 0.50
PIK3CD O00329 2/20 0.50
BTK Q06187 2/20 0.50
BLK P51451 1/20 0.50
BMX P51813 1/20 0.50
JAK3 P52333 1/20 0.50
ERBB4 Q15303 1/20 0.50
VCP P55072 1/20 0.49
KCNH2 Q12809 1/20 0.48
BRAF P15056 2/20 0.47
TNNI3K Q59H18 2/20 0.47
CSF1R P07333 1/20 0.46
ITK Q08881 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21515950 0.91 EGFR (0.51) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20150571 0.90 PIK3CD (0.51) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20139048 0.87 SRC (0.59) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20139083 0.83 EGFR (0.70) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20150708 0.82 PIK3CD (0.54) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20143667 0.82 PIK3CD (0.56) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20138990 0.81 EGFR (0.54) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20138979 0.81 BTK (0.54) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20139788 0.81 PIK3CD (0.49) EGFRSRCFYNERBB2PIK3CD
SCHEMBL20139002 0.80 PIK3CD (0.55) EGFRSRCFYNERBB2PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3556761-A1 PYRROLO-AROMATIC HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF The National Institutes Of Pharmaceutical Research (CN) 2019-10-23 EP disclosed
WO-2018088780-A1 NOVEL PYRROLOPYRIMIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2018-05-17 WO disclosed