SCHEMBL20139083

SCHEMBL20139083

C=CC(=O)Nc1cccc(Nc2ncnc3[nH]c(-c4ccc(Oc5ccccc5)cc4)cc23)c1

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 9/20 0.70
BTK Q06187 9/20 0.70
KCNH2 Q12809 1/20 0.70
ERBB2 P04626 3/20 0.62
SRC P12931 4/20 0.52
FYN P06241 3/20 0.52
VCP P55072 1/20 0.52
PIK3CD O00329 2/20 0.51
BRAF P15056 1/20 0.50
TNNI3K Q59H18 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20139118 0.94 EGFR (0.64) EGFRBTKKCNH2ERBB2SRC
SCHEMBL20138980 0.93 EGFR (0.67) EGFRBTKKCNH2ERBB2SRC
SCHEMBL20139048 0.92 SRC (0.59) EGFRBTKKCNH2ERBB2SRC
SCHEMBL20139002 0.85 PIK3CD (0.55) EGFRBTKKCNH2ERBB2SRC
SCHEMBL20150686 0.83 EGFR (0.50) EGFRBTKKCNH2ERBB2SRC
SCHEMBL20150708 0.83 PIK3CD (0.54) EGFRBTKKCNH2ERBB2SRC
SCHEMBL20143667 0.83 PIK3CD (0.56) EGFRBTKKCNH2ERBB2SRC
SCHEMBL14165496 0.82 BTK (1.00) EGFRBTKKCNH2ERBB2
SCHEMBL20139785 0.82 SRC (0.58) EGFRBTKKCNH2ERBB2SRC
SCHEMBL20138979 0.81 BTK (0.54) EGFRBTKKCNH2ERBB2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018088780-A1 NOVEL PYRROLOPYRIMIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME DAEWOONG PHARMACEUTICAL CO., LTD. (KR) 2018-05-17 WO disclosed