SCHEMBL6919915

SCHEMBL6919915

Cc1nc(-c2cccc(C(=O)N(C)[C@H](CCNC(=O)c3cccn3C)Cc3ccccc3)c2)no1

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.65
HCRTR2 O43614 2/20 0.65
KIFC1 Q9BW19 8/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
DRD3 P35462 2/20 0.38
CTSD P07339 1/20 0.38
HSD11B1 P28845 1/20 0.37
DRD2 P14416 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2013804 0.87 HCRTR1 (0.73) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL6920111 0.86 HCRTR1 (0.68) HCRTR1HCRTR2KIFC1NPC1RAB9A
SCHEMBL2015048 0.85 HCRTR1 (0.72) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL13139093 0.84 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2010792 0.84 HCRTR1 (0.67) HCRTR1HCRTR2NPC1RAB9ADRD3
SCHEMBL13139060 0.83 HCRTR1 (0.77) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2012115 0.83 HCRTR1 (0.65) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2010953 0.83 HCRTR1 (0.69) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2011910 0.83 HCRTR1 (0.69) HCRTR1HCRTR2NPC1RAB9A
SCHEMBL2015121 0.81 HCRTR1 (0.65) HCRTR1HCRTR2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073316-A1 4-ARYL-BUTANE-1,3-DIAMIDES NOVARTIS AG (CH) 2011-06-23 WO disclosed