SCHEMBL20153337

SCHEMBL20153337

N=C(/C=C\N)CCCc1ccc2c(n1)NCCC2

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 17/20 0.51
ITGB3 P05106 14/20 0.51
ITGA2B P08514 1/20 0.50
ITGB6 P18564 9/20 0.46
ITGB5 P18084 6/20 0.46
ITGB8 P26012 6/20 0.46
CXCR4 P61073 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24521901 0.87 ITGAV (0.54) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL23341167 0.83 ITGAV (0.64) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL25636886 0.83 ITGAV (0.63) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL30195434 0.83 ITGAV (0.63) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL24521988 0.80 ITGB3 (0.63) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL5856589 0.80 ITGAV (0.56) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL22029472 0.79 ITGAV (0.68) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL5847742 0.79 ITGAV (0.56) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL13007683 0.78 ITGAV (0.63) ITGAVITGB3ITGA2BITGB6ITGB5
SCHEMBL21340330 0.78 ITGAV (0.60) ITGAVITGB3ITGA2BITGB6ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538525-B1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2022-06-22 EP disclosed
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed