SCHEMBL20153393

SCHEMBL20153393

CCCN[C@@H](CC(=O)OCC)c1ccc(OC)nc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 5/20 0.42
KCNK9 Q9NPC2 1/20 0.41
KMT2A Q03164 5/20 0.40
MEN1 O00255 4/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
OXTR P30559 1/20 0.39
ADRB3 P13945 1/20 0.38
ALDH1A1 P00352 2/20 0.37
POLB P06746 2/20 0.37
PABPC1 P11940 2/20 0.37
THRB P10828 1/20 0.36
P2RX3 P56373 1/20 0.36
P2RX2 Q9UBL9 1/20 0.36
FFAR1 O14842 1/20 0.36
ITGB1 P05556 1/20 0.36
ITGA4 P13612 1/20 0.36
NNMT P40261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23462651 0.91 KCNK3 (0.39) KCNK3KCNK9KMT2AMEN1MAPT
SCHEMBL23558962 0.90 OXTR (0.39) KCNK3KCNK9KMT2AMEN1MAPT
SCHEMBL6108575 0.86 KCNK3 (0.42) KCNK3KCNK9KMT2AMEN1MAPT
SCHEMBL6108573 0.86 KCNK3 (0.42) KCNK3KCNK9KMT2AMEN1MAPT
SCHEMBL20139059 0.81 KCNK3 (0.43) KCNK3KCNK9KMT2AMEN1MAPT
SCHEMBL20141864 0.79 ITGB1 (0.40) KCNK3KCNK9KMT2AMEN1OXTR
SCHEMBL20158341 0.79 KCNK3 (0.39) KCNK3KCNK9MAPTKDM4EOXTR
SCHEMBL6106081 0.79 NNMT (0.43) KCNK3KCNK9KMT2AMEN1MAPT
SCHEMBL20153392 0.79 NNMT (0.43) KCNK3KCNK9KMT2AMEN1MAPT
SCHEMBL6219002 0.78 KMT2A (0.40) KCNK3KCNK9KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018089353-A1 3-SUBSTITUTED PROPIONIC ACIDS AS ALPHA V INTEGRIN INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2018-05-17 WO disclosed