SCHEMBL20154221

SCHEMBL20154221

Cc1nsc(C(=O)OCc2ccccc2)c1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.56
TSHR P16473 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
TDP1 Q9NUW8 4/20 0.50
KMT2A Q03164 3/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A3 Q01959 1/20 0.50
ALDH1A1 P00352 5/20 0.47
LMNA P02545 2/20 0.46
NPC1 O15118 2/20 0.46
MAPT P10636 2/20 0.46
MAPK1 P28482 2/20 0.46
POLB P06746 2/20 0.46
STAT1 P42224 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ATM Q13315 1/20 0.46
HPGD P15428 1/20 0.44
CSNK1D P48730 1/20 0.44
L3MBTL1 Q9Y468 3/20 0.43
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20154222 0.87 RAB9A (0.55) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL20154271 0.80 RAB9A (0.59) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL18924216 0.79 TSHR (0.56) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL22005553 0.77 RAB9A (0.53) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL21550516 0.77 RAB9A (0.71) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL20154269 0.77 RAB9A (0.53) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL20154220 0.77 RAB9A (0.50) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL21572853 0.76 TDP1 (0.58) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL19928470 0.74 TDP1 (0.54) RAB9ATSHRSMN1; SMN2TDP1KMT2A
SCHEMBL20711150 0.73 RAB9A (0.53) RAB9ATSHRSMN1; SMN2TDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3538512-B1 NEW ANTHELMINTIC QUINOLINE-3-CARBOXAMIDE DERIVATIVES BAYER ANIMAL HEALTH GMBH (DE) 2021-06-16 EP disclosed
WO-2021018839-A1 ISOQUINOLINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF PARASITIC INFECTIONS BAYER ANIMAL HEALTH GMBH (DE) 2021-02-04 WO disclosed
WO-2019002132-A1 NEW AZAQUINOLINE DERIVATIVES BAYER ANIMAL HEALTH GMBH (DE) 2019-01-03 WO disclosed
WO-2018087036-A1 NEW ANTHELMINTIC QUINOLINE-3-CARBOXAMIDE DERIVATIVES BAYER ANIMAL HEALTH GMBH (DE) 2018-05-17 WO disclosed