SCHEMBL20154923

SCHEMBL20154923

Cn1cc(Br)c2c(ccn2C)c1=O

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 12/20 0.38
GAA P10253 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
BRD9 Q9H8M2 2/20 0.35
BRD7 Q9NPI1 1/20 0.34
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
CRBN Q96SW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23575586 0.85 BRD4 (0.34) BRD4GAAL3MBTL1BRD9BRD7
SCHEMBL22729417 0.78 BRD4 (0.44) BRD4GAAL3MBTL1BRD9BRD7
SCHEMBL15519363 0.77 GAA (0.37) BRD4GAABRD9CRBN
SCHEMBL16651641 0.72 BRD4 (0.58) BRD4L3MBTL1BRD9BRD7
SCHEMBL29613217 0.72 BRD4 (0.58) BRD4L3MBTL1BRD9BRD7
SCHEMBL20155010 0.71 DGAT1 (0.40)
SCHEMBL17879710 0.71 BRD4 (0.41) BRD4GAAL3MBTL1BRD9BRD7
SCHEMBL17963571 0.70 CCNT1 (0.33) BRD4L3MBTL1
SCHEMBL28520363 0.70 HTT (0.38) BRD4L3MBTL1BRD9
SCHEMBL19657265 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed