SCHEMBL20155010

SCHEMBL20155010

Cn1cc(Br)c2c(ccn2COCC[Si](C)(C)C)c1=O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.40
NPC1 O15118 1/20 0.34
DUT P33316 1/20 0.33
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
EPHB4 P54760 1/20 0.32
TEK Q02763 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15069386 0.90 DGAT1 (0.40) DGAT1NPC1DUTEGFRIGF1R
SCHEMBL1076270 0.81 DGAT1 (0.39) DGAT1NPC1DUT
SCHEMBL30207672 0.78 NPC1 (0.35) DGAT1NPC1DUTEGFRIGF1R
SCHEMBL30902997 0.77 DUT (0.35) DGAT1NPC1DUTEGFRIGF1R
SCHEMBL27214896 0.76 DGAT1 (0.36) DGAT1NPC1
SCHEMBL27233836 0.76 NPC1 (0.42) DGAT1NPC1DUTEGFRIGF1R
SCHEMBL30851323 0.76 NPC1 (0.42) DGAT1NPC1DUTEGFRIGF1R
SCHEMBL25287397 0.75 DGAT1 (0.38) DGAT1NPC1DUTEGFRIGF1R
SCHEMBL20155011 0.75 DGAT1 (0.40) DGAT1NPC1
SCHEMBL21224611 0.75 DGAT1 (0.40) DGAT1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed