SCHEMBL20155098

SCHEMBL20155098

CC/C=C1/c2cn(C)nc2C(c2cc(N)ccc2NCC2CC2)=CN1C

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.35
USP30 Q70CQ3 1/20 0.32
PTGER4 P35408 2/20 0.31
CRHR1 P34998 1/20 0.30
IRAK4 Q9NWZ3 1/20 0.30
TTK P33981 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155507 0.69 BRD4 (0.39) BRD4PTGER4
SCHEMBL20155096 0.66 BRD4 (0.49) BRD4
SCHEMBL20155510 0.64 BRD4 (0.47) BRD4
SCHEMBL27270334 0.62 PTGER4 (0.55) PTGER4CRHR1
SCHEMBL30288293 0.58 USP30 (0.44) BRD4USP30IRAK4TTK
SCHEMBL11935117 0.57 PTGER4 (0.44) BRD4PTGER4
SCHEMBL13438679 0.57 PTGER4 (0.44) BRD4PTGER4
SCHEMBL23610920 0.57 BCL6 (0.49) BRD4PTGER4
SCHEMBL20155486 0.55 ACHE (0.41) BRD4PTGER4
SCHEMBL30288239 0.55 USP30 (0.39) BRD4USP30IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed