SCHEMBL20155486

SCHEMBL20155486

CN1C=C(c2cc([N+](=O)[O-])ccc2NCC2CC2)C(=N)C(=N)C1=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.41
BRD4 O60885 8/20 0.38
PTGER4 P35408 1/20 0.38
CASP1 P29466 1/20 0.37
CASP3 P42574 1/20 0.37
CASP4 P49662 1/20 0.37
CASP7 P55210 1/20 0.37
CASP9 P55211 1/20 0.37
CASP6 P55212 1/20 0.37
ALOX5 P09917 1/20 0.36
ALDH1A1 P00352 4/20 0.35
KMT2A Q03164 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155599 0.88 ACHE (0.37) ACHEBRD4PTGER4CASP1CASP3
SCHEMBL20155507 0.84 BRD4 (0.39) BRD4PTGER4
SCHEMBL20155176 0.75 CASP1 (0.45) ACHECASP1CASP3CASP4CASP7
SCHEMBL14471226 0.72 KAT2B (0.57) PTGER4ALDH1A1KMT2ALMNAMAPT
SCHEMBL23610898 0.70 BCL6 (0.47) ACHEBRD4PTGER4KMT2ALMNA
SCHEMBL30692912 0.70 BCL6 (0.47) ACHEBRD4PTGER4KMT2ALMNA
SCHEMBL28514065 0.69 MAPT (0.55) PTGER4ALDH1A1KMT2ALMNAMAPT
SCHEMBL27267582 0.69 PTGER4 (0.56) PTGER4ALDH1A1KMT2ALMNAMAPT
SCHEMBL20155178 0.68 BRD4 (0.33) BRD4
SCHEMBL14214117 0.67 PTGER4 (0.37) ACHEBRD4PTGER4ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed