SCHEMBL20155102

SCHEMBL20155102

N#Cc1cc(Cl)ccc1Oc1ccc(N)cc1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
ALDH1A1 P00352 3/20 0.47
USP2 O75604 1/20 0.47
MAPT P10636 2/20 0.41
CYP2D6 P10635 2/20 0.41
MEN1 O00255 2/20 0.41
HPGD P15428 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
NOS2 P35228 3/20 0.40
SLC22A12 Q96S37 5/20 0.39
SLC6A2 P23975 4/20 0.38
SLC6A4 P31645 4/20 0.38
MAPK1 P28482 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28688126 0.89 KDM4E (0.59) KDM4EALDH1A1USP2MAPTCYP2D6
SCHEMBL20155143 0.82 ALDH1A1 (0.47) KDM4EALDH1A1USP2SLC22A12MAPK1
SCHEMBL28696921 0.82 KDM4E (0.54) KDM4EALDH1A1USP2MAPTCYP2D6
SCHEMBL29845834 0.80 TTR (0.56) ALDH1A1MAPTMEN1HPGDKMT2A
SCHEMBL28681143 0.79 KDM4E (0.51) KDM4EALDH1A1USP2MAPTCYP2D6
SCHEMBL28678291 0.79 KDM4E (0.55) KDM4EALDH1A1USP2MAPTCYP2D6
SCHEMBL28691780 0.78 KDM4E (0.67) KDM4EALDH1A1USP2MAPTCYP2D6
SCHEMBL29845884 0.77 EPAS1 (0.47) KDM4EALDH1A1MAPTCYP2D6MEN1
SCHEMBL28682193 0.77 KDM4E (0.56) KDM4EALDH1A1USP2MAPTCYP2D6
SCHEMBL20154990 0.77 EPAS1 (0.47) KDM4EALDH1A1MAPTCYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed