SCHEMBL28678291

SCHEMBL28678291

Cc1cc(Cl)ccc1Oc1ccc(N)cc1C#N

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.55
ALDH1A1 P00352 2/20 0.55
USP2 O75604 1/20 0.55
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
HPGD P15428 2/20 0.51
MAPT P10636 2/20 0.48
SLC22A12 Q96S37 2/20 0.47
SLC6A2 P23975 8/20 0.45
SLC6A4 P31645 8/20 0.45
SLC6A3 Q01959 6/20 0.45
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2D6 P10635 1/20 0.44
AR P10275 2/20 0.43
KCNH2 Q12809 2/20 0.41
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28688126 0.89 KDM4E (0.59) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL28696921 0.85 KDM4E (0.54) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL28691780 0.84 KDM4E (0.67) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL28681143 0.82 KDM4E (0.51) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL28682193 0.80 KDM4E (0.56) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL20155102 0.79 KDM4E (0.47) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL28681705 0.79 AR (0.50) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL3356525 0.79 KDM4E (0.50) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL28677203 0.77 AR (0.53) KDM4EALDH1A1USP2MEN1KMT2A
SCHEMBL2033529 0.77 KDM4E (0.56) KDM4EALDH1A1USP2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109651208-B N-aryl sulfonamide compound, pharmaceutical composition and application thereof 中国科学院上海药物研究所 2022-01-04 CN disclosed