SCHEMBL20155138

SCHEMBL20155138

CN/C=C1\C(=N)C(=O)N(C)C=C1c1cc(N)ccc1Nc1ccc(F)cc1F

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.36
BRD4 O60885 4/20 0.34
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PTGS2 P35354 1/20 0.31
ALDH1A1 P00352 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155590 0.92 MAPK14 (0.36) MAPK14BRD4MEN1KMT2APTGS2
SCHEMBL20155146 0.90
SCHEMBL20155062 0.87 MAPK14 (0.39) MAPK14BRD4MEN1KMT2APTGS2
SCHEMBL20155186 0.84 TDO2 (0.31)
SCHEMBL20155038 0.84 BRD4 (0.42) MAPK14BRD4
SCHEMBL20155583 0.83 BRD4 (0.36) BRD4
SCHEMBL20155584 0.83 BRD4 (0.43) BRD4
SCHEMBL20155748 0.82 MAPK14 (0.34) MAPK14BRD4MEN1KMT2AHSD17B10
SCHEMBL20155483 0.81 MAPK14 (0.37) MAPK14BRD4MEN1KMT2APTGS2
SCHEMBL20155635 0.80 MAPK14 (0.33) MAPK14BRD4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed