SCHEMBL20155748

SCHEMBL20155748

CON/C=C1\C(=N)C(c2cc(N)ccc2Nc2ccc(F)cc2F)=CN(C)C1=O

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.34
BRD4 O60885 3/20 0.32
HSD17B10 Q99714 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20155635 0.90 MAPK14 (0.33) MAPK14BRD4HSD17B10
SCHEMBL20155590 0.90 MAPK14 (0.36) MAPK14BRD4HSD17B10MEN1KMT2A
SCHEMBL20155483 0.86 MAPK14 (0.37) MAPK14BRD4MEN1KMT2A
SCHEMBL20155068 0.85 BRD4 (0.41) MAPK14BRD4
SCHEMBL20155062 0.84 MAPK14 (0.39) MAPK14BRD4HSD17B10MEN1KMT2A
SCHEMBL20155138 0.82 MAPK14 (0.36) MAPK14BRD4HSD17B10MEN1KMT2A
SCHEMBL20155186 0.81 TDO2 (0.31)
SCHEMBL20155650 0.78 AKT1 (0.31) MAPK14BRD4
SCHEMBL20155291 0.76 BRD4 (0.42) MAPK14BRD4
SCHEMBL20155621 0.76 MAPK14 (0.34) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086604-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATIONS THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed